BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 3 hits Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase' and Ligand = 'BDBM510496'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Tyrosine-protein kinase


(Dog)
BDBM510496
PNG
(US11077111, Compound IVa | US20230295171, Example ...)
Show SMILES Cn1cc(cn1)-c1nc(N[C@@H]2CCCC[C@@H]2N)c(Cl)c2CNC(=O)c12
PDB

UniProtKB/TrEMBL

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 323n/an/an/an/an/an/a


TBA

Assay Description
A radiometric protein kinase assay was used for measuring the kinase activity of the Dog (Canis lupus familiaris) IRAK4, JAK1, JAK2, SYK kinases. All...


Citation and Details

BindingDB Entry DOI: 10.7270/Q2K35XS9
More data for this
Ligand-Target Pair
Tyrosine-protein kinase


(Dog)
BDBM510496
PNG
(US11077111, Compound IVa | US20230295171, Example ...)
Show SMILES Cn1cc(cn1)-c1nc(N[C@@H]2CCCC[C@@H]2N)c(Cl)c2CNC(=O)c12
PDB

UniProtKB/TrEMBL

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 466n/an/an/an/an/an/a


TBA

Assay Description
A radiometric protein kinase assay was used for measuring the kinase activity of the Dog (Canis lupus familiaris) IRAK4, JAK1, JAK2, SYK kinases. All...


Citation and Details

BindingDB Entry DOI: 10.7270/Q2K35XS9
More data for this
Ligand-Target Pair
Tyrosine-protein kinase


(Dog)
BDBM510496
PNG
(US11077111, Compound IVa | US20230295171, Example ...)
Show SMILES Cn1cc(cn1)-c1nc(N[C@@H]2CCCC[C@@H]2N)c(Cl)c2CNC(=O)c12
PDB

UniProtKB/TrEMBL

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 624n/an/an/an/an/an/a


TBA

Assay Description
A radiometric protein kinase assay was used for measuring the kinase activity of the Dog (Canis lupus familiaris) IRAK4, JAK1, JAK2, SYK kinases. All...


Citation and Details

BindingDB Entry DOI: 10.7270/Q2K35XS9
More data for this
Ligand-Target Pair