Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tyrosine-protein kinase ABL1 (Homo sapiens (Human)) | BDBM50252767 ((2'Z-3'E)-6-Bromoindirubin-3'-[O-(2-{4-[2-(2-hydro...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
Beckman Research Institute Curated by ChEMBL | Assay Description Inhibitory constant against Serotonin transporter | J Nat Prod 79: 2464-2471 (2016) Article DOI: 10.1021/acs.jnatprod.6b00285 BindingDB Entry DOI: 10.7270/Q2GF0WZR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase ABL1 (Homo sapiens (Human)) | BDBM50252767 ((2'Z-3'E)-6-Bromoindirubin-3'-[O-(2-{4-[2-(2-hydro...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 34.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Beckman Research Institute Curated by ChEMBL | Assay Description Inhibition of recombinant ABL1 (unknown origin) after 120 mins in presence of [33P]ATP | J Nat Prod 79: 2464-2471 (2016) Article DOI: 10.1021/acs.jnatprod.6b00285 BindingDB Entry DOI: 10.7270/Q2GF0WZR | |||||||||||
More data for this Ligand-Target Pair |