Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Vasopressin V1a receptor (Homo sapiens (Human)) | BDBM50052954![]() (2-Methyl-N-[4-(2,3,4,5-tetrahydro-benzo[b]azepine-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 8.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UMR7200 CNRS/Universit£ de Strasbourg Curated by ChEMBL | Assay Description Binding affinity to vasopressin V1a receptor | J Med Chem 55: 8588-602 (2012) Article DOI: 10.1021/jm3006146 BindingDB Entry DOI: 10.7270/Q28G8MT5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vasopressin V1a receptor (RAT) | BDBM50052954![]() (2-Methyl-N-[4-(2,3,4,5-tetrahydro-benzo[b]azepine-...) | UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 56 | n/a | n/a | n/a | n/a | n/a | n/a |
Otsuka Pharmaceutical Co. Curated by ChEMBL | Assay Description Displacement of [3H]-AVP from AVP-V1a receptor binding site in rat liver | J Med Chem 39: 3547-55 (1996) Article DOI: 10.1021/jm960133o BindingDB Entry DOI: 10.7270/Q2DZ07CT | |||||||||||
More data for this Ligand-Target Pair |