Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Voltage-dependent T-type calcium channel subunit alpha-1G (Homo sapiens (Human)) | BDBM50543609 (CHEMBL4647557) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyung Hee University Curated by ChEMBL | Assay Description Inhibition of human Cav3.1 expressed in tsA-201 cells by patch clamp electrophysiology | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2020.115491 BindingDB Entry DOI: 10.7270/Q2NC64R3 | |||||||||||
More data for this Ligand-Target Pair |