Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
cAMP-dependent protein kinase catalytic subunit alpha/beta/gamma (Homo sapiens (Human)) | BDBM50287090![]() (4-Chloro-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of the platelet-derived growth factor receptor. | Bioorg Med Chem Lett 7: 187-192 (1997) Article DOI: 10.1016/S0960-894X(96)00601-4 BindingDB Entry DOI: 10.7270/Q23X86MF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cAMP-dependent protein kinase catalytic subunit alpha/beta/gamma (Homo sapiens (Human)) | BDBM50287090![]() (4-Chloro-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of serine/threonine kinase(PKA) | Bioorg Med Chem Lett 6: 1221-1226 (1996) Article DOI: 10.1016/0960-894X(96)00197-7 BindingDB Entry DOI: 10.7270/Q2348KBG | |||||||||||
More data for this Ligand-Target Pair |