BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'cGMP-dependent protein kinase' and Ligand = 'BDBM340886'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
cGMP-dependent protein kinase


()		BDBM340886
PNG
(1-cyclopentyl-3-(naphthalen-1-ylmethyl)-1H- pyrazo...)
Show SMILES Nc1ncnc2n(nc(Cc3cccc4ccccc34)c12)C1CCCC1
Show InChI InChI=1S/C21H21N5/c22-20-19-18(12-15-8-5-7-14-6-1-4-11-17(14)15)25-26(16-9-2-3-10-16)21(19)24-13-23-20/h1,4-8,11,13,16H,2-3,9-10,12H2,(H2,22,23,24)
UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 553n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...

Citation and Details

BindingDB Entry DOI: 10.7270/Q2K077GQ
More data for this
Ligand-Target Pair