Compile Data Set for Download or QSAR

Found 35 hits Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50012172   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554960 (CHEMBL4749555) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccc(cc1C(F)(F)F)C#N)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554959 (CHEMBL4797312) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccc(Cl)cc1C(F)(F)F)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	7.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554970 (CHEMBL4784771) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1cc(ccc1N)C#N |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	19	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554971 (CHEMBL4763693) Show SMILES COc1ccc(cc1OC[C@@H](N)CCNS(=O)(=O)c1ccc(Cl)cc1Cl)C#N |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	28	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554972 (CHEMBL4755223) Show SMILES Cc1ccc(cc1OC[C@@H](N)CCNS(=O)(=O)c1ccc(Cl)cc1Cl)C#N |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	40	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554957 (CHEMBL4795311) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccccc1C(F)(F)F)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	40	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554973 (CHEMBL4761250) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1cc(ccc1F)C#N |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	42	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554945 (CHEMBL4753854) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	50	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554974 (CHEMBL4777668) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1cc(ccc1Cl)C#N |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	58	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554964 (CHEMBL4740898) Show SMILES NC(CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1cccc(c1)C#N Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	63	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554958 (CHEMBL4747177) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccccc1[N+]([O-])=O)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	63	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50450502 (CHEMBL3218112) Show SMILES OC1(COc2ccc(C#N)c(F)c2)CCN(CC1)S(=O)(=O)c1ccc(Cl)cc1Cl Show InChI InChI=1S/C19H17Cl2FN2O4S/c20-14-2-4-18(16(21)9-14)29(26,27)24-7-5-19(25,6-8-24)12-28-15-3-1-13(11-23)17(22)10-15/h1-4,9-10,25H,5-8,12H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	100	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554942 (CHEMBL4749498) Show SMILES NC(CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1ccc(C#N)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	126	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554963 (CHEMBL4787004) Show SMILES NC(CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1ccc(cc1)C#N Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	200	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554961 (CHEMBL4754934) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccc(cc1Cl)C(F)(F)F)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	316	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554956 (CHEMBL4800371) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccccc1OC(F)(F)F)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	631	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554951 (CHEMBL4788545) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccc(cc1)C(F)(F)F)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	631	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554941 (CHEMBL4741577) Show SMILES OC(CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1ccc(C#N)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	794	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554952 (CHEMBL4765224) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccc(cc1)C#N)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	794	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554966 (CHEMBL4784636) Show SMILES NC(CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1cccc(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554954 (CHEMBL4741595) Show SMILES Cc1ccccc1S(=O)(=O)NCC[C@H](N)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554946 (CHEMBL4746378) Show SMILES N[C@H](CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554948 (CHEMBL4740502) Show SMILES NC(CCNS(=O)(=O)c1ccccc1Cl)COc1ccc(C#N)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.26E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554962 (CHEMBL4747398) Show SMILES NC(CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.59E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554955 (CHEMBL4757902) Show SMILES N[C@@H](CCNS(=O)(=O)c1ccccc1-c1ccccc1)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554944 (CHEMBL4797224) Show SMILES CN(CCC(N)COc1ccc(C#N)c(F)c1)S(=O)(=O)c1ccc(Cl)cc1Cl Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.51E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554965 (CHEMBL4782089) Show SMILES NC(CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1ccccc1C#N Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.51E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554950 (CHEMBL4790603) Show SMILES NC(CCNS(=O)(=O)c1ccc(Cl)cc1)COc1ccc(C#N)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.01E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554969 (CHEMBL4751191) Show SMILES COc1cccc(OCC(N)CCNS(=O)(=O)c2ccc(Cl)cc2Cl)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	6.31E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554953 (CHEMBL4789107) Show SMILES COc1ccccc1S(=O)(=O)NCC[C@H](N)COc1ccc(C#N)c(F)c1 |r| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	7.94E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554943 (CHEMBL4745283) Show SMILES CN(CCC(O)COc1ccc(C#N)c(F)c1)S(=O)(=O)c1ccc(Cl)cc1Cl Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554967 (CHEMBL4794809) Show SMILES NC(CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1cccc(Cl)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.26E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554949 (CHEMBL4788203) Show SMILES NC(CCNS(=O)(=O)c1cccc(Cl)c1)COc1ccc(C#N)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.26E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554947 (CHEMBL4799509) Show SMILES NC(CCNS(=O)(=O)c1ccccc1)COc1ccc(C#N)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human))	BDBM50554968 (CHEMBL4744266) Show SMILES Cc1cccc(OCC(N)CCNS(=O)(=O)c2ccc(Cl)cc2Cl)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	<2.51E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...				Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01303 BindingDB Entry DOI: 10.7270/Q2XW4PFK
					More data for this Ligand-Target Pair