Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Orexin receptor type 2 (Homo sapiens (Human)) | BDBM50434481![]() (CHEMBL2385132 | CHEMBL2385133 | CHEMBL2385134) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | PDB Article PubMed | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School Curated by ChEMBL | Assay Description Antagonist activity at OX2 receptor (unknown origin) | Bioorg Med Chem Lett 23: 3389-92 (2013) Article DOI: 10.1016/j.bmcl.2013.03.079 BindingDB Entry DOI: 10.7270/Q279461B | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Orexin receptor type 2 (Homo sapiens (Human)) | BDBM50434481![]() (CHEMBL2385132 | CHEMBL2385133 | CHEMBL2385134) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School Curated by ChEMBL | Assay Description Antagonist activity at OX2 receptor (unknown origin) | Bioorg Med Chem Lett 23: 3389-92 (2013) Article DOI: 10.1016/j.bmcl.2013.03.079 BindingDB Entry DOI: 10.7270/Q279461B | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) |