Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase N1 (Homo sapiens (Human)) | BDBM50399676 (CHEMBL2178352 | US9096601, 8-26) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 6.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sichuan University Curated by ChEMBL | Assay Description Inhibition of human recombinant PKN1 by radiometric kinase assay | J Med Chem 55: 10685-99 (2012) Article DOI: 10.1021/jm301365e BindingDB Entry DOI: 10.7270/Q2251KBV | |||||||||||
More data for this Ligand-Target Pair |