Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM25759![]() (CHEMBL723 | Carvedilol | Coreg | Dilatrend | Eucar...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet ![]() | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Rzesz£w University of Technology Curated by ChEMBL | Assay Description Displacement of [3H]Prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membrane by liquid scintillation counting | Eur J Med Chem 44: 5103-11 (2009) Article DOI: 10.1016/j.ejmech.2009.07.012 BindingDB Entry DOI: 10.7270/Q2668H17 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50480959![]() (CHEMBL573951) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Rzesz£w University of Technology Curated by ChEMBL | Assay Description Displacement of [3H]Prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membrane by liquid scintillation counting | Eur J Med Chem 44: 5103-11 (2009) Article DOI: 10.1016/j.ejmech.2009.07.012 BindingDB Entry DOI: 10.7270/Q2668H17 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50480955![]() (CHEMBL573946) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Rzesz£w University of Technology Curated by ChEMBL | Assay Description Displacement of [3H]Prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membrane by liquid scintillation counting | Eur J Med Chem 44: 5103-11 (2009) Article DOI: 10.1016/j.ejmech.2009.07.012 BindingDB Entry DOI: 10.7270/Q2668H17 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50480956![]() (CHEMBL572571) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 46 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Rzesz£w University of Technology Curated by ChEMBL | Assay Description Displacement of [3H]Prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membrane by liquid scintillation counting | Eur J Med Chem 44: 5103-11 (2009) Article DOI: 10.1016/j.ejmech.2009.07.012 BindingDB Entry DOI: 10.7270/Q2668H17 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50480958![]() (CHEMBL582863) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 61 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Rzesz£w University of Technology Curated by ChEMBL | Assay Description Displacement of [3H]Prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membrane by liquid scintillation counting | Eur J Med Chem 44: 5103-11 (2009) Article DOI: 10.1016/j.ejmech.2009.07.012 BindingDB Entry DOI: 10.7270/Q2668H17 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50480957![]() (CHEMBL574593) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 76 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Rzesz£w University of Technology Curated by ChEMBL | Assay Description Displacement of [3H]Prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membrane by liquid scintillation counting | Eur J Med Chem 44: 5103-11 (2009) Article DOI: 10.1016/j.ejmech.2009.07.012 BindingDB Entry DOI: 10.7270/Q2668H17 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50267196![]() ((+/-)1-(1H-indol-4-yloxy)-3-(2-(2-methoxyphenoxy)e...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Rzesz£w University of Technology Curated by ChEMBL | Assay Description Displacement of [3H]Prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membrane by liquid scintillation counting | Eur J Med Chem 44: 5103-11 (2009) Article DOI: 10.1016/j.ejmech.2009.07.012 BindingDB Entry DOI: 10.7270/Q2668H17 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50480954![]() (CHEMBL573945) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 169 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Rzesz£w University of Technology Curated by ChEMBL | Assay Description Displacement of [3H]Prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membrane by liquid scintillation counting | Eur J Med Chem 44: 5103-11 (2009) Article DOI: 10.1016/j.ejmech.2009.07.012 BindingDB Entry DOI: 10.7270/Q2668H17 | |||||||||||
More data for this Ligand-Target Pair |