Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human)) | BDBM50126022 (CHEMBL26512 | {[3-(Biphenyl-4-yloxy)-3-(4-fluoro-p...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Binding affinity towards rat hippocampus GlyT1 transporter expressed in HEK 293 cells | Bioorg Med Chem Lett 13: 1291-2 (2003) BindingDB Entry DOI: 10.7270/Q2JM291Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent glycine transporter 1 (Homo sapiens (Human)) | BDBM50126023 ((Methyl-{3-[4-(4-methyl-benzoyl)-phenoxy]-3-phenyl...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Binding affinity towards rat hippocampus GlyT1 transporter expressed in HEK 293 cells | Bioorg Med Chem Lett 13: 1291-2 (2003) BindingDB Entry DOI: 10.7270/Q2JM291Q | |||||||||||
More data for this Ligand-Target Pair |