Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50008175 (4-(8-Aza-spiro[4.5]dec-8-ylcarbamoyl)-4-(3-chloro-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Rotta Research Laboratorium Curated by ChEMBL | Assay Description Concentration required to inhibit by 50% the specific binding of [3H]pentagastrin to Cholecystokinin type B receptor in rabbit gastric gland | J Med Chem 35: 28-38 (1992) BindingDB Entry DOI: 10.7270/Q2XS5W11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50008202 (4-(3,5-Dichloro-benzoylamino)-4-(3,3-dimethyl-buty...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rotta Research Laboratorium Curated by ChEMBL | Assay Description Concentration required to inhibit by 50% the specific binding of [3H]pentagastrin to Cholecystokinin type B receptor in rabbit gastric gland | J Med Chem 35: 28-38 (1992) BindingDB Entry DOI: 10.7270/Q2XS5W11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50008184 (4-(3-Chloro-benzoylamino)-4-(3,3-dimethyl-butylcar...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rotta Research Laboratorium Curated by ChEMBL | Assay Description Concentration required to inhibit by 50% the specific binding of [3H]pentagastrin to Cholecystokinin type B receptor in rabbit gastric gland | J Med Chem 35: 28-38 (1992) BindingDB Entry DOI: 10.7270/Q2XS5W11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50008163 (4-(2-Adamantan-1-yl-ethylcarbamoyl)-4-(3,5-dichlor...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rotta Research Laboratorium Curated by ChEMBL | Assay Description Concentration required to inhibit by 50% the specific binding of [3H]pentagastrin to Cholecystokinin type B receptor in rabbit gastric gland | J Med Chem 35: 28-38 (1992) BindingDB Entry DOI: 10.7270/Q2XS5W11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50008190 (4-(2-Adamantan-1-yl-ethylcarbamoyl)-4-(3-chloro-be...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rotta Research Laboratorium Curated by ChEMBL | Assay Description Concentration required to inhibit by 50% the specific binding of [3H]pentagastrin to Cholecystokinin type B receptor in rabbit gastric gland | J Med Chem 35: 28-38 (1992) BindingDB Entry DOI: 10.7270/Q2XS5W11 | |||||||||||
More data for this Ligand-Target Pair |