Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Corticotropin-releasing factor receptor 1 (Rattus norvegicus (rat)) | BDBM50403726![]() (CHEMBL2112936) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
A Subsidiary of Agouron Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 1 | Bioorg Med Chem Lett 9: 765-70 (1999) BindingDB Entry DOI: 10.7270/Q2TD9WJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Corticotropin-releasing factor receptor 1 (Rattus norvegicus (rat)) | BDBM50075917![]() (8N-(2-aminoethyl)-15-oxo-9a,10,11,12,13,13a,14,15-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 160 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
A Subsidiary of Agouron Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 1 | Bioorg Med Chem Lett 9: 765-70 (1999) BindingDB Entry DOI: 10.7270/Q2TD9WJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Corticotropin-releasing factor receptor 1 (Rattus norvegicus (rat)) | BDBM50075918![]() (8N-[2-amino-(1R,2R)-cyclohexyl]-15-oxo-(9aS,13aS)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 180 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
A Subsidiary of Agouron Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 1 | Bioorg Med Chem Lett 9: 765-70 (1999) BindingDB Entry DOI: 10.7270/Q2TD9WJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Corticotropin-releasing factor receptor 1 (Rattus norvegicus (rat)) | BDBM50403725![]() (CHEMBL2112326) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
A Subsidiary of Agouron Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 1 | Bioorg Med Chem Lett 9: 765-70 (1999) BindingDB Entry DOI: 10.7270/Q2TD9WJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Corticotropin-releasing factor receptor 1 (Rattus norvegicus (rat)) | BDBM50075921![]() (8N-(2-aminoethyl)-15-oxo-(9aR,13aS)-11,12,13,15-te...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 270 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
A Subsidiary of Agouron Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 1 | Bioorg Med Chem Lett 9: 765-70 (1999) BindingDB Entry DOI: 10.7270/Q2TD9WJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Corticotropin-releasing factor receptor 1 (Rattus norvegicus (rat)) | BDBM50075924![]() (13-Oxo-10,11,12,13-tetrahydro-9H-5,7,9,12-tetraaza...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
A Subsidiary of Agouron Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 1 | Bioorg Med Chem Lett 9: 765-70 (1999) BindingDB Entry DOI: 10.7270/Q2TD9WJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Corticotropin-releasing factor receptor 1 (Rattus norvegicus (rat)) | BDBM50075920![]() (7-Oxo-7H-benzo[e]perimidine-4-carboxylic acid ((1R...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
A Subsidiary of Agouron Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 1 | Bioorg Med Chem Lett 9: 765-70 (1999) BindingDB Entry DOI: 10.7270/Q2TD9WJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Corticotropin-releasing factor receptor 1 (Rattus norvegicus (rat)) | BDBM50075923![]() (7-Oxo-7H-benzo[e]perimidine-4-carboxylic acid ((1R...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
A Subsidiary of Agouron Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 1 | Bioorg Med Chem Lett 9: 765-70 (1999) BindingDB Entry DOI: 10.7270/Q2TD9WJJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Corticotropin-releasing factor receptor 1 (Rattus norvegicus (rat)) | BDBM50075919![]() (7-Oxo-7H-benzo[e]perimidine-4-carboxylic acid (2-a...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
A Subsidiary of Agouron Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 1 | Bioorg Med Chem Lett 9: 765-70 (1999) BindingDB Entry DOI: 10.7270/Q2TD9WJJ | |||||||||||
More data for this Ligand-Target Pair |