Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Phenylalanine--tRNA ligase alpha/beta subunit (Haemophilus influenzae) | BDBM18116 (2-[2-({[(2R)-2-(4-bromothiophen-2-yl)-2-hydroxyeth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 56 | n/a | n/a | n/a | n/a | 2.0 | n/a |
GSK | Assay Description The reactions were performed in 96-well Packard 384-well Packard Optiplates. After 10 min of incubation, the reaction was stopped by addition of a co... | Bioorg Med Chem Lett 15: 2305-9 (2005) Article DOI: 10.1016/j.bmcl.2005.03.003 BindingDB Entry DOI: 10.7270/Q25D8Q3C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phenylalanine--tRNA ligase alpha/beta subunit (Haemophilus influenzae) | BDBM18103 (2-({[2-(1H-1,3-benzodiazol-2-ylmethoxy)phenyl]meth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | 2.0 | n/a |
GSK | Assay Description The reactions were performed in 96-well Packard 384-well Packard Optiplates. After 10 min of incubation, the reaction was stopped by addition of a co... | Bioorg Med Chem Lett 15: 2305-9 (2005) Article DOI: 10.1016/j.bmcl.2005.03.003 BindingDB Entry DOI: 10.7270/Q25D8Q3C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phenylalanine--tRNA ligase alpha/beta subunit (Haemophilus influenzae) | BDBM18117 (2-[2-({[(2S)-2-(4-bromothiophen-2-yl)-2-hydroxyeth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | 2.0 | n/a |
GSK | Assay Description The reactions were performed in 96-well Packard 384-well Packard Optiplates. After 10 min of incubation, the reaction was stopped by addition of a co... | Bioorg Med Chem Lett 15: 2305-9 (2005) Article DOI: 10.1016/j.bmcl.2005.03.003 BindingDB Entry DOI: 10.7270/Q25D8Q3C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phenylalanine--tRNA ligase alpha/beta subunit (Haemophilus influenzae) | BDBM18098 (2-({[2-(benzyloxy)phenyl]methyl}amino)-1-(4-bromot...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | 7.9 | 37 |
GSK | Assay Description The reactions were performed in 96-well Packard 384-well Packard Optiplates. After 10 min of incubation, the reaction was stopped by addition of a co... | Bioorg Med Chem Lett 15: 2305-9 (2005) Article DOI: 10.1016/j.bmcl.2005.03.003 BindingDB Entry DOI: 10.7270/Q25D8Q3C | |||||||||||
More data for this Ligand-Target Pair |