Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM50482687 (CHEMBL426916) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Wuhan Institute of Technology Curated by ChEMBL | Assay Description Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptor | Eur J Med Chem 45: 3595-600 (2010) Article DOI: 10.1016/j.ejmech.2010.05.004 BindingDB Entry DOI: 10.7270/Q27D2XZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM50482692 (CHEMBL390326) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Wuhan Institute of Technology Curated by ChEMBL | Assay Description Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptor | Eur J Med Chem 45: 3595-600 (2010) Article DOI: 10.1016/j.ejmech.2010.05.004 BindingDB Entry DOI: 10.7270/Q27D2XZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238234 (US9388210, 14a | US9388210, 6a) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238243 (US9388210, 16a) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 28 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM50482694 (CHEMBL229535) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Wuhan Institute of Technology Curated by ChEMBL | Assay Description Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptor | Eur J Med Chem 45: 3595-600 (2010) Article DOI: 10.1016/j.ejmech.2010.05.004 BindingDB Entry DOI: 10.7270/Q27D2XZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM50482688 (CHEMBL387958) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Wuhan Institute of Technology Curated by ChEMBL | Assay Description Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptor | Eur J Med Chem 45: 3595-600 (2010) Article DOI: 10.1016/j.ejmech.2010.05.004 BindingDB Entry DOI: 10.7270/Q27D2XZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM50215531 (2-chloro-alpha-[[(4-chlorophenyl)amino]methylene]-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Wuhan Institute of Technology Curated by ChEMBL | Assay Description Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptor | Eur J Med Chem 45: 3595-600 (2010) Article DOI: 10.1016/j.ejmech.2010.05.004 BindingDB Entry DOI: 10.7270/Q27D2XZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM50482691 (CHEMBL556727) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
Wuhan Institute of Technology Curated by ChEMBL | Assay Description Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptor | Eur J Med Chem 45: 3595-600 (2010) Article DOI: 10.1016/j.ejmech.2010.05.004 BindingDB Entry DOI: 10.7270/Q27D2XZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM50482690 (CHEMBL229374) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Wuhan Institute of Technology Curated by ChEMBL | Assay Description Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptor | Eur J Med Chem 45: 3595-600 (2010) Article DOI: 10.1016/j.ejmech.2010.05.004 BindingDB Entry DOI: 10.7270/Q27D2XZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238245 (US9388210, 17a) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 53 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238238 (US9388210, 13a | US9388210, 15a) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 56 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM50482696 (CHEMBL229201) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 79 | n/a | n/a | n/a | n/a | n/a | n/a |
Wuhan Institute of Technology Curated by ChEMBL | Assay Description Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptor | Eur J Med Chem 45: 3595-600 (2010) Article DOI: 10.1016/j.ejmech.2010.05.004 BindingDB Entry DOI: 10.7270/Q27D2XZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238234 (US9388210, 14a | US9388210, 6a) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 128 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM50482686 (CHEMBL227018) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 158 | n/a | n/a | n/a | n/a | n/a | n/a |
Wuhan Institute of Technology Curated by ChEMBL | Assay Description Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptor | Eur J Med Chem 45: 3595-600 (2010) Article DOI: 10.1016/j.ejmech.2010.05.004 BindingDB Entry DOI: 10.7270/Q27D2XZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM50482689 (CHEMBL388639) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 398 | n/a | n/a | n/a | n/a | n/a | n/a |
Wuhan Institute of Technology Curated by ChEMBL | Assay Description Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptor | Eur J Med Chem 45: 3595-600 (2010) Article DOI: 10.1016/j.ejmech.2010.05.004 BindingDB Entry DOI: 10.7270/Q27D2XZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238238 (US9388210, 13a | US9388210, 15a) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 474 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238235 (US9388210, 14b | US9388210, 6b) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 501 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238244 (US9388210, 16b) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 544 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238246 (US9388210, 17b) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 605 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238236 (US9388210, 6c) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 629 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238248 (US9388210, 5b) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 770 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238247 (US9388210, 5a) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 997 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238249 (US9388210, 5c) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.02E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238239 (US9388210, 13b | US9388210, 15b) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM50482695 (CHEMBL227017) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wuhan Institute of Technology Curated by ChEMBL | Assay Description Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptor | Eur J Med Chem 45: 3595-600 (2010) Article DOI: 10.1016/j.ejmech.2010.05.004 BindingDB Entry DOI: 10.7270/Q27D2XZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238237 (US9388210, 6d) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.84E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238235 (US9388210, 14b | US9388210, 6b) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.03E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM50482693 (CHEMBL388638) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wuhan Institute of Technology Curated by ChEMBL | Assay Description Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptor | Eur J Med Chem 45: 3595-600 (2010) Article DOI: 10.1016/j.ejmech.2010.05.004 BindingDB Entry DOI: 10.7270/Q27D2XZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 (Rattus norvegicus (Rat)) | BDBM238239 (US9388210, 13b | US9388210, 15b) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 9.60E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
WASHINGTON UNIVERSITY US Patent | Assay Description Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−... | US Patent US9388210 (2016) BindingDB Entry DOI: 10.7270/Q29K4949 | |||||||||||
More data for this Ligand-Target Pair |