Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2 (Homo sapiens (Human)) | BDBM50445605 (CHEMBL3104001) | PDB UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 690 | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr... | Bioorg Med Chem Lett 24: 674-8 (2014) Article DOI: 10.1016/j.bmcl.2013.11.049 BindingDB Entry DOI: 10.7270/Q2RF5WH9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2 (Homo sapiens (Human)) | BDBM50445612 (CHEMBL3103985) | PDB UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 700 | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr... | Bioorg Med Chem Lett 24: 674-8 (2014) Article DOI: 10.1016/j.bmcl.2013.11.049 BindingDB Entry DOI: 10.7270/Q2RF5WH9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2 (Homo sapiens (Human)) | BDBM50445611 (CHEMBL3103988) | PDB UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 790 | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr... | Bioorg Med Chem Lett 24: 674-8 (2014) Article DOI: 10.1016/j.bmcl.2013.11.049 BindingDB Entry DOI: 10.7270/Q2RF5WH9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2 (Homo sapiens (Human)) | BDBM50445610 (CHEMBL3104068) | PDB UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr... | Bioorg Med Chem Lett 24: 674-8 (2014) Article DOI: 10.1016/j.bmcl.2013.11.049 BindingDB Entry DOI: 10.7270/Q2RF5WH9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2 (Homo sapiens (Human)) | BDBM50445609 (CHEMBL3103999) | PDB UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr... | Bioorg Med Chem Lett 24: 674-8 (2014) Article DOI: 10.1016/j.bmcl.2013.11.049 BindingDB Entry DOI: 10.7270/Q2RF5WH9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2 (Homo sapiens (Human)) | BDBM50445608 (CHEMBL3104126) | PDB UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr... | Bioorg Med Chem Lett 24: 674-8 (2014) Article DOI: 10.1016/j.bmcl.2013.11.049 BindingDB Entry DOI: 10.7270/Q2RF5WH9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2 (Homo sapiens (Human)) | BDBM50445607 (CHEMBL3104079) | PDB UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr... | Bioorg Med Chem Lett 24: 674-8 (2014) Article DOI: 10.1016/j.bmcl.2013.11.049 BindingDB Entry DOI: 10.7270/Q2RF5WH9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2 (Homo sapiens (Human)) | BDBM50445606 (CHEMBL3103983) | PDB UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr... | Bioorg Med Chem Lett 24: 674-8 (2014) Article DOI: 10.1016/j.bmcl.2013.11.049 BindingDB Entry DOI: 10.7270/Q2RF5WH9 | |||||||||||
More data for this Ligand-Target Pair |