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Compile Data Set for Download or QSAR

Found 1 hit of ec50 for UniProtKB: P48039   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melatonin receptor type 1A/1B


(Homo sapiens (Human))		BDBM50149182
PNG
(CHEMBL124577 | N-[3-(2-Methyl-benzooxazol-7-yl)-pr...)
Show SMILES CCC(=O)NCCCc1cccc2nc(C)oc12
Show InChI InChI=1S/C14H18N2O2/c1-3-13(17)15-9-5-7-11-6-4-8-12-14(11)18-10(2)16-12/h4,6,8H,3,5,7,9H2,1-2H3,(H,15,17)
PDB

KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
antibodypedia
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/an/an/a 0.260n/an/an/an/a



Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Agonist activity for its ability to inhibit forskolin-stimulated cAMP accumulation against MT1 receptor

Bioorg Med Chem Lett 14: 3799-802 (2004)


Article DOI: 10.1016/j.bmcl.2004.04.082
BindingDB Entry DOI: 10.7270/Q2S75FSR
More data for this
Ligand-Target Pair