Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Pyruvate dehydrogenase E1 component subunit alpha,/beta, mitochondrial (Pisum sativum) | BDBM50486217 (CLACYFOS) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.28E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central China Normal University Curated by ChEMBL | Assay Description Inhibition of PDHc in Vigna radiata var. radiata VC2778A shoot mitochondria assessed as decrease in rate of NADH formation using sodium pyruvate as s... | J Agric Food Chem 59: 4801-13 (2011) Article DOI: 10.1021/jf104247w BindingDB Entry DOI: 10.7270/Q2V69NFJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate dehydrogenase E1 component subunit alpha,/beta, mitochondrial (Pisum sativum) | BDBM50486218 (CHEMBL2227928) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.97E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central China Normal University Curated by ChEMBL | Assay Description Inhibition of PDHc in Vigna radiata var. radiata VC2778A shoot mitochondria assessed as decrease in rate of NADH formation using sodium pyruvate as s... | J Agric Food Chem 59: 4801-13 (2011) Article DOI: 10.1021/jf104247w BindingDB Entry DOI: 10.7270/Q2V69NFJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate dehydrogenase E1 component subunit alpha,/beta, mitochondrial (Pisum sativum) | BDBM50486214 (CHEMBL2227973) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.31E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central China Normal University Curated by ChEMBL | Assay Description Inhibition of PDHc in Vigna radiata var. radiata VC2778A shoot mitochondria assessed as decrease in rate of NADH formation using sodium pyruvate as s... | J Agric Food Chem 59: 4801-13 (2011) Article DOI: 10.1021/jf104247w BindingDB Entry DOI: 10.7270/Q2V69NFJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate dehydrogenase E1 component subunit alpha,/beta, mitochondrial (Pisum sativum) | BDBM50486215 (CHEMBL2227682) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.54E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central China Normal University Curated by ChEMBL | Assay Description Inhibition of PDHc in Vigna radiata var. radiata VC2778A shoot mitochondria assessed as decrease in rate of NADH formation using sodium pyruvate as s... | J Agric Food Chem 59: 4801-13 (2011) Article DOI: 10.1021/jf104247w BindingDB Entry DOI: 10.7270/Q2V69NFJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pyruvate dehydrogenase E1 component subunit alpha,/beta, mitochondrial (Pisum sativum) | BDBM50486213 ((2,4-Dichlorophenoxy)Acetic Acid | 2,4-Dichlorophe...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >4.53E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Central China Normal University Curated by ChEMBL | Assay Description Inhibition of PDHc in Pisum sativum Zhongwan-2 (pea) shoot mitochondria assessed as decrease in rate of NADH formation using sodium pyruvate as subst... | J Agric Food Chem 59: 4801-13 (2011) Article DOI: 10.1021/jf104247w BindingDB Entry DOI: 10.7270/Q2V69NFJ | |||||||||||
More data for this Ligand-Target Pair |