Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Mu-type opioid/Nociceptin receptor (Rattus norvegicus (rat)-RAT) | BDBM50492400 (CHEMBL2403214) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 316 | n/a | n/a | n/a | n/a |
Bulgarian Academy of Sciences Curated by ChEMBL | Assay Description Activity at Wistar rat NOP/mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction | Bioorg Med Chem Lett 23: 4052-5 (2013) Article DOI: 10.1016/j.bmcl.2013.05.064 BindingDB Entry DOI: 10.7270/Q2639SNZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid/Nociceptin receptor (Rattus norvegicus (rat)-RAT) | BDBM50492403 (CHEMBL2403213) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 550 | n/a | n/a | n/a | n/a |
Bulgarian Academy of Sciences Curated by ChEMBL | Assay Description Activity at Wistar rat NOP/mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of... | Bioorg Med Chem Lett 23: 4052-5 (2013) Article DOI: 10.1016/j.bmcl.2013.05.064 BindingDB Entry DOI: 10.7270/Q2639SNZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid/Nociceptin receptor (Rattus norvegicus (rat)-RAT) | BDBM50492400 (CHEMBL2403214) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 617 | n/a | n/a | n/a | n/a |
Bulgarian Academy of Sciences Curated by ChEMBL | Assay Description Activity at Wistar rat NOP/mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of... | Bioorg Med Chem Lett 23: 4052-5 (2013) Article DOI: 10.1016/j.bmcl.2013.05.064 BindingDB Entry DOI: 10.7270/Q2639SNZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid/Nociceptin receptor (Rattus norvegicus (rat)-RAT) | BDBM50492403 (CHEMBL2403213) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.66E+3 | n/a | n/a | n/a | n/a |
Bulgarian Academy of Sciences Curated by ChEMBL | Assay Description Activity at Wistar rat NOP/mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction | Bioorg Med Chem Lett 23: 4052-5 (2013) Article DOI: 10.1016/j.bmcl.2013.05.064 BindingDB Entry DOI: 10.7270/Q2639SNZ | |||||||||||
More data for this Ligand-Target Pair |