Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tubulin alpha chain-like 3/1A chain/1B chain/1C chain/3C chain/3E chain/4A chain/8 chain (Human-Homo sapiens) | BDBM50517652 (CHEMBL4584084) | PDB MMDB UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 540 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Curated by ChEMBL | Assay Description Inhibition of tubulin alpha in human A2780 cells assessed as reduction in cell growth | J Med Chem 62: 1684-1689 (2019) Article DOI: 10.1021/acs.jmedchem.8b01774 BindingDB Entry DOI: 10.7270/Q24X5C5V | |||||||||||
More data for this Ligand-Target Pair |