BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 4 hits of ki for UniProtKB: P30937   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Somatostatin receptor type 1/2/3/4/5


(RAT)
BDBM50214420
PNG
(CHEMBL330352)
Show SMILES NCCCCCN1c2ccccc2CN(C(Cc2c[nH]c3ccccc23)C1=O)C(=O)c1ccccc1
Show InChI InChI=1S/C30H32N4O2/c31-17-9-2-10-18-33-27-16-8-5-13-23(27)21-34(29(35)22-11-3-1-4-12-22)28(30(33)36)19-24-20-32-26-15-7-6-14-25(24)26/h1,3-8,11-16,20,28,32H,2,9-10,17-19,21,31H2
PDB
MMDB

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars

6.30E+3n/an/an/an/an/an/an/an/a


TBA

Assay Description
Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligand


Citation and Details

BindingDB Entry DOI: 10.7270/Q20G3NBX
More data for this
Ligand-Target Pair
Somatostatin receptor type 1/2/3/4/5


(RAT)
BDBM50214420
PNG
(CHEMBL330352)
Show SMILES NCCCCCN1c2ccccc2CN(C(Cc2c[nH]c3ccccc23)C1=O)C(=O)c1ccccc1
Show InChI InChI=1S/C30H32N4O2/c31-17-9-2-10-18-33-27-16-8-5-13-23(27)21-34(29(35)22-11-3-1-4-12-22)28(30(33)36)19-24-20-32-26-15-7-6-14-25(24)26/h1,3-8,11-16,20,28,32H,2,9-10,17-19,21,31H2
PDB
MMDB

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars

6.30E+3n/an/an/an/an/an/an/an/a


TBA

Assay Description
Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligand


Citation and Details

BindingDB Entry DOI: 10.7270/Q20G3NBX
More data for this
Ligand-Target Pair
Somatostatin receptor type 1/2/3/4/5


(RAT)
BDBM50214420
PNG
(CHEMBL330352)
Show SMILES NCCCCCN1c2ccccc2CN(C(Cc2c[nH]c3ccccc23)C1=O)C(=O)c1ccccc1
Show InChI InChI=1S/C30H32N4O2/c31-17-9-2-10-18-33-27-16-8-5-13-23(27)21-34(29(35)22-11-3-1-4-12-22)28(30(33)36)19-24-20-32-26-15-7-6-14-25(24)26/h1,3-8,11-16,20,28,32H,2,9-10,17-19,21,31H2
PDB
MMDB

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars

6.31E+3n/an/an/an/an/an/an/an/a


TBA

Assay Description
Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligand


Citation and Details

BindingDB Entry DOI: 10.7270/Q20G3NBX
More data for this
Ligand-Target Pair
Somatostatin receptor type 1/2/3/4/5


(RAT)
BDBM50212468
PNG
(CHEMBL28415)
Show SMILES NCCCCCOCC1OC(OCCc2c[nH]c3ccccc23)C(OCc2ccccc2)C1OCc1ccccc1
Show InChI InChI=1S/C34H42N2O5/c35-19-10-3-11-20-37-25-31-32(39-23-26-12-4-1-5-13-26)33(40-24-27-14-6-2-7-15-27)34(41-31)38-21-18-28-22-36-30-17-9-8-16-29(28)30/h1-2,4-9,12-17,22,31-34,36H,3,10-11,18-21,23-25,35H2
PDB
MMDB

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars

1.86E+4n/an/an/an/an/an/an/an/a


TBA

Assay Description
Inhibitory activity against Somatostatin receptor in rat cortex membrane using 125 I-Tyrs-octreotide as radioligand


Citation and Details

BindingDB Entry DOI: 10.7270/Q2X350M0
More data for this
Ligand-Target Pair