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Compile Data Set for Download or QSAR

Found 1 hit of ec50 for monomerid = 50017656   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histamine H1 receptor


(Cavia porcellus (domestic guinea pig))		BDBM50017656
PNG
(CHEMBL1193 | Dimethyl-(3-phenyl-3-pyridin-2-yl-pro...)
Show SMILES CN(C)CCC(c1ccccc1)c1ccccn1
Show InChI InChI=1S/C16H20N2/c1-18(2)13-11-15(14-8-4-3-5-9-14)16-10-6-7-12-17-16/h3-10,12,15H,11,13H2,1-2H3
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Article
PubMed
n/an/an/an/a 2.82E+4n/an/an/an/a



Cairo University

Curated by ChEMBL


Assay Description
Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced contractions at 5 ug/ml

Bioorg Med Chem 16: 9009-17 (2008)


Article DOI: 10.1016/j.bmc.2008.08.039
BindingDB Entry DOI: 10.7270/Q2PR7ZSZ
More data for this
Ligand-Target Pair