Compile Data Set for Download or QSAR

Found 2 hits of ec50 for monomerid = 50103562   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50103562 (CHEMBL3357995) Show SMILES C[C@@H]1CN(CCN1c1ncc(OCc2ccc(cc2C#N)S(C)(=O)=O)cn1)c1nnc(o1)C(F)(F)F |r| Show InChI InChI=1S/C21H20F3N7O4S/c1-13-11-30(20-29-28-18(35-20)21(22,23)24)5-6-31(13)19-26-9-16(10-27-19)34-12-14-3-4-17(36(2,32)33)7-15(14)8-25/h3-4,7,9-10,13H,5-6,11-12H2,1-2H3/t13-/m1/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	55	n/a	n/a	n/a	n/a
AstraZeneca Curated by ChEMBL					Assay Description Agonist activity at human GPR119 expressed in HEK293S cells assessed as cAMP accumulation incubated for 45 mins by HTRF assay				J Med Chem 57: 8984-98 (2014) Article DOI: 10.1021/jm5011012 BindingDB Entry DOI: 10.7270/Q29G5PK1
					More data for this Ligand-Target Pair
Glucose-dependent insulinotropic receptor (Mus musculus)	BDBM50103562 (CHEMBL3357995) Show SMILES C[C@@H]1CN(CCN1c1ncc(OCc2ccc(cc2C#N)S(C)(=O)=O)cn1)c1nnc(o1)C(F)(F)F |r| Show InChI InChI=1S/C21H20F3N7O4S/c1-13-11-30(20-29-28-18(35-20)21(22,23)24)5-6-31(13)19-26-9-16(10-27-19)34-12-14-3-4-17(36(2,32)33)7-15(14)8-25/h3-4,7,9-10,13H,5-6,11-12H2,1-2H3/t13-/m1/s1	Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	1.98E+3	n/a	n/a	n/a	n/a
AstraZeneca Curated by ChEMBL					Assay Description Agonist activity at mouse GPR119 expressed in HEK293S cells assessed as cAMP accumulation incubated for 45 mins by HTRF assay				J Med Chem 57: 8984-98 (2014) Article DOI: 10.1021/jm5011012 BindingDB Entry DOI: 10.7270/Q29G5PK1
					More data for this Ligand-Target Pair