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Compile Data Set for Download or QSAR

Found 1 hit of ec50 for monomerid = 50140887   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Period circadian protein homolog 2


(Homo sapiens (Human))		BDBM50140887
PNG
(CHEMBL3753709)
Show SMILES OC(CN1CCS1(=O)=O)Cn1c2ccccc2c2ccccc12
Show InChI InChI=1S/C17H18N2O3S/c20-13(11-18-9-10-23(18,21)22)12-19-16-7-3-1-5-14(16)15-6-2-4-8-17(15)19/h1-8,13,20H,9-12H2
PDB

UniProtKB/SwissProt

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PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/an/an/a 190n/an/an/an/a



Reset Therapeutics

Curated by ChEMBL


Assay Description
Reduction of amplitude effect of PER2 in human U2OS cells harboring Per2-dLuc luciferase reporter gene assessed as effects on circadian rhythms

Bioorg Med Chem Lett 26: 757-60 (2016)


Article DOI: 10.1016/j.bmcl.2015.12.102
BindingDB Entry DOI: 10.7270/Q2DR2XCS
More data for this
Ligand-Target Pair