Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50165940 (Ac-YRC(Me)*EHdFRWC(Me)NH2 | CHEMBL427666) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.920 | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at human Melanocortin-4 receptor as peptide required for 50% maximal cAMP release (n > or =2) | J Med Chem 48: 3095-8 (2005) Article DOI: 10.1021/jm0501432 BindingDB Entry DOI: 10.7270/Q2251HQZ | |||||||||||
More data for this Ligand-Target Pair |