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Compile Data Set for Download or QSAR

Found 1 hit of ec50 for monomerid = 50326222   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Muscarinic acetylcholine receptor M1


(Homo sapiens (Human))		BDBM50326222
PNG
(CHEMBL1243295 | Cyclobutanecarboxylic acid{1-[3-(3...)
Show SMILES O=C(NC1CCN(CCCN2C(=O)COc3ccccc23)CC1)C1CCC1
Show InChI InChI=1S/C21H29N3O3/c25-20-15-27-19-8-2-1-7-18(19)24(20)12-4-11-23-13-9-17(10-14-23)22-21(26)16-5-3-6-16/h1-2,7-8,16-17H,3-6,9-15H2,(H,22,26)
UniProtKB/SwissProt

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Similars
Article
PubMed
n/an/an/an/a 160n/an/an/an/a



H. Lundbeck A/S

Curated by ChEMBL


Assay Description
Agonist activity at human muscarinic M1 receptor expressed in CHO-K1 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assay

J Med Chem 53: 6386-97 (2010)


Article DOI: 10.1021/jm100697g
BindingDB Entry DOI: 10.7270/Q2765G9K
More data for this
Ligand-Target Pair