Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bombesin receptor subtype-3 (Homo sapiens (Human)) | BDBM50394613 (CHEMBL2164580) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assay | ACS Med Chem Lett 3: 252-256 (2012) Article DOI: 10.1021/ml200304j BindingDB Entry DOI: 10.7270/Q2PG1ST9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50394613 (CHEMBL2164580) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 57 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assay | ACS Med Chem Lett 3: 252-256 (2012) Article DOI: 10.1021/ml200304j BindingDB Entry DOI: 10.7270/Q2PG1ST9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 1 group I member 2 (Homo sapiens (Human)) | BDBM50394613 (CHEMBL2164580) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.18E+4 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Activation of PXR | ACS Med Chem Lett 3: 252-256 (2012) Article DOI: 10.1021/ml200304j BindingDB Entry DOI: 10.7270/Q2PG1ST9 | |||||||||||
More data for this Ligand-Target Pair |