Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50400776 (CHEMBL2204986) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 19 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at GPR119 in human HEK293 cells assessed as cAMP level by beta-lactamase reporter gene assay | ACS Med Chem Lett 3: 955-958 (2012) Article DOI: 10.1021/ml300296q BindingDB Entry DOI: 10.7270/Q2SB46WV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50400776 (CHEMBL2204986) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 30 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at GPR119 in human U20S cells assessed as binding to beta-arrestin by chemilumiscence analysis | ACS Med Chem Lett 3: 955-958 (2012) Article DOI: 10.1021/ml300296q BindingDB Entry DOI: 10.7270/Q2SB46WV | |||||||||||
More data for this Ligand-Target Pair |