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Compile Data Set for Download or QSAR

Found 1 hit of ec50 for monomerid = 50542061   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Atypical chemokine receptor 3


(Homo sapiens (Human))		BDBM50542061
PNG
(CHEMBL4634148)
Show SMILES NC(=O)C([C@@H]1CCN(CCOc2ccc(cc2)-c2nccs2)C1)(c1ccccc1)c1ccccc1 |r|
Show InChI InChI=1S/C29H29N3O2S/c30-28(33)29(23-7-3-1-4-8-23,24-9-5-2-6-10-24)25-15-17-32(21-25)18-19-34-26-13-11-22(12-14-26)27-31-16-20-35-27/h1-14,16,20,25H,15,17-19,21H2,(H2,30,33)/t25-/m1/s1
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a>1.00E+4n/an/an/an/a



Pfizer Inc.

Curated by ChEMBL


Assay Description
Agonist activity at human CXCR7 receptor expressed in CHOK1 cell membranes assessed as increase in beta-arrestin recruitment incubated for 30 mins

ACS Med Chem Lett 11: 1330-1334 (2020)


Article DOI: 10.1021/acsmedchemlett.0c00163
BindingDB Entry DOI: 10.7270/Q2J38X4M
More data for this
Ligand-Target Pair