Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Microtubule-associated protein tau (Homo sapiens (Human)) | BDBM50020859 (CHEMBL3286982) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Temple University School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of recombinant human microtubule associated protein tau aggregation by Thiazin-red R displacement fluorescence assay | ACS Med Chem Lett 5: 619-20 (2014) Article DOI: 10.1021/ml500147n BindingDB Entry DOI: 10.7270/Q2ZW1NGS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amyloid-beta precursor protein (Homo sapiens (Human)) | BDBM50020859 (CHEMBL3286982) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
Temple University School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of amyloid beta (unknown origin) aggregation by Thiazin-red R displacement fluorescence assay | ACS Med Chem Lett 5: 619-20 (2014) Article DOI: 10.1021/ml500147n BindingDB Entry DOI: 10.7270/Q2ZW1NGS | |||||||||||
More data for this Ligand-Target Pair |