Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50046145 (2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.85E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd. Curated by ChEMBL | Assay Description Inhibition of rat CPT1A using [3H]carnitine by radiometric assay | J Med Chem 54: 3109-52 (2011) Article DOI: 10.1021/jm100809g BindingDB Entry DOI: 10.7270/Q29K4CDQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 1, liver isoform (Rattus norvegicus) | BDBM50046145 (2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.85E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd. Curated by ChEMBL | Assay Description Inhibition of rat CPT1A using [3H]carnitine by radiometric assay | J Med Chem 54: 3109-52 (2011) Article DOI: 10.1021/jm100809g BindingDB Entry DOI: 10.7270/Q29K4CDQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 2, mitochondrial (Rattus norvegicus) | BDBM50046145 (2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.75E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd. Curated by ChEMBL | Assay Description Inhibition of rat CPT2 using [3H]carnitine by radiometric assay | J Med Chem 54: 3109-52 (2011) Article DOI: 10.1021/jm100809g BindingDB Entry DOI: 10.7270/Q29K4CDQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carnitine O-palmitoyltransferase 2, mitochondrial (Rattus norvegicus) | BDBM50046145 (2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.75E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd. Curated by ChEMBL | Assay Description Inhibition of rat CPT2 using [3H]carnitine by radiometric assay | J Med Chem 54: 3109-52 (2011) Article DOI: 10.1021/jm100809g BindingDB Entry DOI: 10.7270/Q29K4CDQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C zeta type (Rattus norvegicus) | BDBM50046145 (2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 4.96E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Louisiana State University Curated by ChEMBL | Assay Description Inhibition of protein kinase C (PKC) purified from rat brain | J Med Chem 36: 177-8 (1993) BindingDB Entry DOI: 10.7270/Q2Z321VQ | |||||||||||
More data for this Ligand-Target Pair |