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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50060151   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha


(Rattus norvegicus-Rattus norvegicus (rat))		BDBM50060151
PNG
(CHEMBL408134 | [(S)-1-{(4-Benzyloxy-benzyl)-[(1,1-...)
Show SMILES CC(C)(Cc1ccccc1)NC(=O)CN(Cc1ccc(OCc2ccccc2)cc1)C(=O)[C@H](Cc1cnc[nH]1)NC(=O)OCc1ccccc1
Show InChI InChI=1S/C40H43N5O5/c1-40(2,23-30-12-6-3-7-13-30)44-37(46)26-45(25-31-18-20-35(21-19-31)49-27-32-14-8-4-9-15-32)38(47)36(22-34-24-41-29-42-34)43-39(48)50-28-33-16-10-5-11-17-33/h3-21,24,29,36H,22-23,25-28H2,1-2H3,(H,41,42)(H,43,48)(H,44,46)/t36-/m0/s1
PDB

KEGG

UniProtKB/SwissProt

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AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/a 270n/an/an/an/an/an/a



Warner-Lambert Company

Curated by ChEMBL


Assay Description
In vitro inhibition of rat farnesyltransferase.

J Med Chem 40: 3319-22 (1997)


Article DOI: 10.1021/jm970470c
BindingDB Entry DOI: 10.7270/Q2V69HQG
More data for this
Ligand-Target Pair