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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50108882   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Nuclear receptor ROR-gamma


(Homo sapiens (Human))		BDBM50108882
PNG
(CHEMBL3596593)
Show SMILES Cc1ccc(cc1-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl)C(N)=O
Show InChI InChI=1S/C24H20ClFN2O2/c1-14-7-8-17(23(27)29)13-18(14)15-9-10-21-16(12-15)4-3-11-28(21)24(30)22-19(25)5-2-6-20(22)26/h2,5-10,12-13H,3-4,11H2,1H3,(H2,27,29)
PDB

UniProtKB/SwissProt

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PC sid
UniChem

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Article
PubMed
n/an/a 300n/an/an/an/an/an/a



Biogen Idec Inc.

Curated by ChEMBL


Assay Description
Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...

Bioorg Med Chem Lett 25: 2991-7 (2015)


Article DOI: 10.1016/j.bmcl.2015.05.026
BindingDB Entry DOI: 10.7270/Q2ZP47XQ
More data for this
Ligand-Target Pair