Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Prostaglandin D2 receptor 2 (Homo sapiens (Human)) | BDBM50161748 (CHEMBL194085 | [3-((R)-4-Fluoro-benzenesulfonylami...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
7TM Pharma A/S Curated by ChEMBL | Assay Description Inhibition of PGD2-induced inositol phosphate formation at human chemoattractant receptor-homologous molecule expressed on TH2 cells | J Med Chem 48: 897-900 (2005) Article DOI: 10.1021/jm049036i BindingDB Entry DOI: 10.7270/Q24J0DMD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin D2 receptor 2 (Homo sapiens (Human)) | BDBM50161748 (CHEMBL194085 | [3-((R)-4-Fluoro-benzenesulfonylami...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
7TM Pharma A/S Curated by ChEMBL | Assay Description Inhibition of beta-arrestin translocation at human chemoattractant receptor-homologous molecule expressed on TH2 cells in BRET assay | J Med Chem 48: 897-900 (2005) Article DOI: 10.1021/jm049036i BindingDB Entry DOI: 10.7270/Q24J0DMD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (Homo sapiens (Human)) | BDBM50161748 (CHEMBL194085 | [3-((R)-4-Fluoro-benzenesulfonylami...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
7TM Pharma A/S Curated by ChEMBL | Assay Description Inhibition of U-46,619-induced inositol phosphate accumulation at human Thromboxane A2 receptor | J Med Chem 48: 897-900 (2005) Article DOI: 10.1021/jm049036i BindingDB Entry DOI: 10.7270/Q24J0DMD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin D2 receptor (Homo sapiens (Human)) | BDBM50161748 (CHEMBL194085 | [3-((R)-4-Fluoro-benzenesulfonylami...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
7TM Pharma A/S Curated by ChEMBL | Assay Description Inhibition of [3H]-PGD-2 binding to human Prostaglandin D2 receptor | J Med Chem 48: 897-900 (2005) Article DOI: 10.1021/jm049036i BindingDB Entry DOI: 10.7270/Q24J0DMD | |||||||||||
More data for this Ligand-Target Pair |