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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50264012   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histamine H3 receptor


(Homo sapiens (Human))		BDBM50264012
PNG
(4-(4-chlorophenyl)-N-methyl-N-(2-(piperidin-1-yl)e...)
Show SMILES CN(CCN1CCCCC1)C(=O)N1CCN(CC1)c1ccc(Cl)cc1
Show InChI InChI=1S/C19H29ClN4O/c1-21(11-12-22-9-3-2-4-10-22)19(25)24-15-13-23(14-16-24)18-7-5-17(20)6-8-18/h5-8H,2-4,9-16H2,1H3
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Similars
Article
PubMed
n/an/a 160n/an/an/an/an/an/a



Tsukuba Research Institute

Curated by ChEMBL


Assay Description
Inverse agonist activity at human cloned histamine H3 receptor assessed as inhibition of (R)-alpha-methylhistamine-induced [35S]GTPgammaS binding

Bioorg Med Chem Lett 18: 5101-6 (2008)


Article DOI: 10.1016/j.bmcl.2008.07.125
BindingDB Entry DOI: 10.7270/Q2PC3268
More data for this
Ligand-Target Pair