Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Endothelin-1 receptor (Mus musculus) | BDBM50281579 ((S)-3-{2-[((R)-2-Acetylamino-3-phenyl-propionyl)-b...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50281579 ((S)-3-{2-[((R)-2-Acetylamino-3-phenyl-propionyl)-b...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description The inhibitory constant of the compound was evaluated against Endothelin A receptor | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair |