Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Substance-P receptor (GUINEA PIG) | BDBM50283253 ((S)-2-[2-((S)-2-{(S)-2-[(S)-2-((S)-2-Acetylamino-4...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Concentration producing half-maximal inhibition of specific binding of. [125I]-Bolton-Hunter Substance P to NK-1 receptors in the guinea pig cerebral... | Bioorg Med Chem Lett 4: 2263-2266 (1994) Article DOI: 10.1016/0960-894X(94)85022-4 BindingDB Entry DOI: 10.7270/Q2959HHG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuromedin-K receptor (GUINEA PIG) | BDBM50283253 ((S)-2-[2-((S)-2-{(S)-2-[(S)-2-((S)-2-Acetylamino-4...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 533 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Concentration producing half-maximal inhibition of specific binding of [3H]-Senktide to Tachykinin receptor 3 in the guinea pig cerebral cortex | Bioorg Med Chem Lett 4: 2263-2266 (1994) Article DOI: 10.1016/0960-894X(94)85022-4 BindingDB Entry DOI: 10.7270/Q2959HHG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50283253 ((S)-2-[2-((S)-2-{(S)-2-[(S)-2-((S)-2-Acetylamino-4...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 637 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Concentration producing half-maximal inhibition of specific binding of. [125I]-Neurokinin A to NK-2 receptors in the hamster urinary bladder | Bioorg Med Chem Lett 4: 2263-2266 (1994) Article DOI: 10.1016/0960-894X(94)85022-4 BindingDB Entry DOI: 10.7270/Q2959HHG | |||||||||||
More data for this Ligand-Target Pair |