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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50401093   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Metabotropic glutamate receptor 3


(Homo sapiens (Human))		BDBM50401093
PNG
(CHEMBL2204443)
Show SMILES COc1ccc(cc1)C#Cc1ccc(cc1)C(=O)N1CCN(CC1)C(C)C
Show InChI InChI=1S/C23H26N2O2/c1-18(2)24-14-16-25(17-15-24)23(26)21-10-6-19(7-11-21)4-5-20-8-12-22(27-3)13-9-20/h6-13,18H,14-17H2,1-3H3
PDB

UniProtKB/SwissProt

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CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a



Vanderbilt University Medical Center

Curated by ChEMBL


Assay Description
Negative allosteric modulation of mGlu3 assessed as thaillium flux through GIRK channels by cell-based assay

Bioorg Med Chem Lett 22: 3921-5 (2012)


Article DOI: 10.1016/j.bmcl.2012.04.112
BindingDB Entry DOI: 10.7270/Q21N828X
More data for this
Ligand-Target Pair