Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Lethal(3)malignant brain tumor-like protein 3 (Homo sapiens (Human)) | BDBM50440607 (CHEMBL2426375) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lethal(3)malignant brain tumor-like protein 3 (Homo sapiens (Human)) | BDBM50440607 (CHEMBL2426375) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of L3MBTL3 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lethal(3)malignant brain tumor-like protein 4 (Homo sapiens (Human)) | BDBM50440607 (CHEMBL2426375) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of L3MBTL4 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
MBT domain-containing protein 1 (Homo sapiens (Human)) | BDBM50440607 (CHEMBL2426375) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of MBTD1 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4) (Homo sapiens (Human)) | BDBM50440607 (CHEMBL2426375) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of L3MBTL1 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
E3 ubiquitin-protein ligase UHRF1 (Homo sapiens (Human)) | BDBM50440607 (CHEMBL2426375) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of UHRF1 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TP53-binding protein 1 (Homo sapiens (Human)) | BDBM50440607 (CHEMBL2426375) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50440607 (CHEMBL2426375) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PHD finger protein 23 (Homo sapiens (Human)) | BDBM50440607 (CHEMBL2426375) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of PHF23 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Scm-like with four MBT domains protein 1 (Homo sapiens (Human)) | BDBM50440607 (CHEMBL2426375) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of SFMBT1 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysine-specific demethylase 5A (Homo sapiens (Human)) | BDBM50440607 (CHEMBL2426375) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of JARID1A (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair |