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Compile Data Set for Download or QSAR

Found 1 hit of ki for monomerid = 258755   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1 [E4Q,A5T]


(Homo sapiens (Human))		BDBM258755
PNG
(US9499482, 154)
Show SMILES COc1cc(ccc1OCCN1CCC2(COC2)CC1)N1CC=C(Oc2ccc(cc2)C2CC2)C1=O |t:25|
Show InChI InChI=1S/C29H34N2O5/c1-33-27-18-23(6-9-25(27)35-17-16-30-14-11-29(12-15-30)19-34-20-29)31-13-10-26(28(31)32)36-24-7-4-22(5-8-24)21-2-3-21/h4-10,18,21H,2-3,11-17,19-20H2,1H3
UniProtKB/SwissProt

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PC cid
PC sid
UniChem
US Patent
 0.5n/an/an/an/an/an/a7.4n/a



Bristol-Myers Squibb Company

US Patent


Assay Description
An in vitro binding assay was used to determine the compound Ki value or ability to antagonize binding of a peptide agonist to the human melanin conc...

US Patent US9499482 (2016)


BindingDB Entry DOI: 10.7270/Q2M907KT
More data for this
Ligand-Target Pair