Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 (Homo sapiens (Human)) | BDBM50035612 (CHEMBL96926 | OCTANOIC ACID [3S-[3ALPHA, 3ABETA, 4...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | MMDB PDB Article PubMed | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of SERCA1a (unknown origin) ATPase activity | Citation and Details Article DOI: 10.1016/j.bmcl.2017.12.050 BindingDB Entry DOI: 10.7270/Q2KD21HX | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |