Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
B2 bradykinin receptor (Cavia porcellus) | BDBM50045213 (CHEMBL2370042 | D-Arg-Arg-Pro-Hyp-N-methylGly-Phe-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Scios Nova Inc. Curated by ChEMBL | Assay Description Binding affinity against [3H]-bradykinin binding to bradykinin receptor B2 in guinea pig ileal membrane | J Med Chem 36: 2569-71 (1993) BindingDB Entry DOI: 10.7270/Q25D8QX4 | |||||||||||
More data for this Ligand-Target Pair |