Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Translocator protein (Rattus norvegicus (rat)) | BDBM50159084 (CHEMBL179459 | N-Butyl-2-[6,8-dichloro-2-(4-chloro...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Bari Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from peripheral benzodiazepine receptor of rat cerebral cortex | J Med Chem 48: 292-305 (2005) Article DOI: 10.1021/jm049610q BindingDB Entry DOI: 10.7270/Q2RR1XQ0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50159084 (CHEMBL179459 | N-Butyl-2-[6,8-dichloro-2-(4-chloro...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Bari Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from peripheral benzodiazepine receptor of rat ovary | J Med Chem 48: 292-305 (2005) Article DOI: 10.1021/jm049610q BindingDB Entry DOI: 10.7270/Q2RR1XQ0 | |||||||||||
More data for this Ligand-Target Pair |