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Compile Data Set for Download or QSAR

Found 1 hit of ki for monomerid = 50270059   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Furin


(Homo sapiens (Human))		BDBM50270059
PNG
(CHEMBL506175 | TPRARRRKKRD)
Show SMILES [#6]-[#6@@H](-[#8])-[#6@H](-[#7])-[#6](=O)-[#7]-1-[#6]-[#6]-[#6]-[#6@H]-1-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6](-[#8])=O)-[#6](-[#7])=O |r|
Show InChI InChI=1S/C58H111N29O14/c1-30(78-45(93)34(15-7-23-73-54(63)64)85-52(100)40-20-12-28-87(40)53(101)42(61)31(2)88)44(92)79-35(16-8-24-74-55(65)66)48(96)82-37(18-10-26-76-57(69)70)50(98)83-36(17-9-25-75-56(67)68)49(97)81-32(13-3-5-21-59)46(94)80-33(14-4-6-22-60)47(95)84-38(19-11-27-77-58(71)72)51(99)86-39(43(62)91)29-41(89)90/h30-40,42,88H,3-29,59-61H2,1-2H3,(H2,62,91)(H,78,93)(H,79,92)(H,80,94)(H,81,97)(H,82,96)(H,83,98)(H,84,95)(H,85,100)(H,86,99)(H,89,90)(H4,63,64,73)(H4,65,66,74)(H4,67,68,75)(H4,69,70,76)(H4,71,72,77)/t30-,31+,32-,33-,34-,35-,36-,37-,38-,39-,40-,42-/m0/s1
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Article
PubMed
 56n/an/an/an/an/an/an/an/a



Institute for Medical Research

Curated by ChEMBL


Assay Description
Inhibition of human recombinant furin assessed as fluorescent Pyr-RTKR-AMC substrate cleavage

J Biol Chem 282: 20847-53 (2007)


Article DOI: 10.1074/jbc.M703847200
BindingDB Entry DOI: 10.7270/Q2057FPB
More data for this
Ligand-Target Pair