Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50302765 (CHEMBL569755 | N,N-diethyl-4-((3-hydroxyphenyl)(1-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.420 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca R&D Montr£al Curated by ChEMBL | Assay Description Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptor | Bioorg Med Chem Lett 19: 5994-8 (2009) Article DOI: 10.1016/j.bmcl.2009.09.072 BindingDB Entry DOI: 10.7270/Q22J6BX8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50302765 (CHEMBL569755 | N,N-diethyl-4-((3-hydroxyphenyl)(1-...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 88 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca R&D Montr£al Curated by ChEMBL | Assay Description Displacement of [125I]FK33824 from human cloned mu opioid receptor | Bioorg Med Chem Lett 19: 5994-8 (2009) Article DOI: 10.1016/j.bmcl.2009.09.072 BindingDB Entry DOI: 10.7270/Q22J6BX8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50302765 (CHEMBL569755 | N,N-diethyl-4-((3-hydroxyphenyl)(1-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 744 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca R&D Montr£al Curated by ChEMBL | Assay Description Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptor | Bioorg Med Chem Lett 19: 5994-8 (2009) Article DOI: 10.1016/j.bmcl.2009.09.072 BindingDB Entry DOI: 10.7270/Q22J6BX8 | |||||||||||
More data for this Ligand-Target Pair |