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Compile Data Set for Download or QSAR

Found 1 hit of ki for monomerid = 50395752   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Growth hormone secretagogue receptor type 1


(Homo sapiens (Human))		BDBM50395752
PNG
(CHEMBL2164500)
Show SMILES Clc1cc2NC(=O)C(NC(=O)CN3CCN(CC=C)CC3)(c2c(Cl)c1)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C23H22Cl4N4O2/c1-2-5-30-6-8-31(9-7-30)13-20(32)29-23(14-3-4-16(25)17(26)10-14)21-18(27)11-15(24)12-19(21)28-22(23)33/h2-4,10-12H,1,5-9,13H2,(H,28,33)(H,29,32)
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Article
PubMed
 121n/an/an/an/an/an/an/an/a



Sanofi Research

Curated by ChEMBL


Assay Description
Displacement of [125I]-ghrelin from human GHSR1 expressed in CHO-CREluc cells after 1 hr by scintillation counting

Bioorg Med Chem 20: 5623-36 (2012)


Article DOI: 10.1016/j.bmc.2012.07.018
BindingDB Entry DOI: 10.7270/Q2HD7WS4
More data for this
Ligand-Target Pair