Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50543752 (CHEMBL4640400) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 6.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Siena Curated by ChEMBL | Assay Description Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in HEK cell membrane | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2020.115513 BindingDB Entry DOI: 10.7270/Q2R49VB2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50543752 (CHEMBL4640400) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Siena Curated by ChEMBL | Assay Description Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in HEK cell membrane | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2020.115513 BindingDB Entry DOI: 10.7270/Q2R49VB2 | |||||||||||
More data for this Ligand-Target Pair |