Found 10 hits of ic50 for monomerid = 34142 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
5-hydroxytryptamine receptor 4
(GUINEA PIG) | BDBM34142
(2-ethyl-5-methoxy-N,N-dimethyltryptamine | CHEMBL2...)Show InChI InChI=1S/C15H22N2O/c1-5-14-12(8-9-17(2)3)13-10-11(18-4)6-7-15(13)16-14/h6-7,10,16H,5,8-9H2,1-4H3 | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
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CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsson Research AB
Curated by ChEMBL
| Assay Description Inhibitory activity against 5-hydroxytryptamine 4 receptor in guinea pig |
Bioorg Med Chem Lett 15: 4230-4 (2005)
Article DOI: 10.1016/j.bmcl.2005.06.067 BindingDB Entry DOI: 10.7270/Q2ZG6RST |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 6
(Homo sapiens (Human)) | BDBM34142
(2-ethyl-5-methoxy-N,N-dimethyltryptamine | CHEMBL2...)Show InChI InChI=1S/C15H22N2O/c1-5-14-12(8-9-17(2)3)13-10-11(18-4)6-7-15(13)16-14/h6-7,10,16H,5,8-9H2,1-4H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 85 | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsson Research AB
Curated by ChEMBL
| Assay Description Displacement of [3H]-LSD binding to cloned human 5-hydroxytryptamine 6 receptor stably expressed in HEK cells |
Bioorg Med Chem Lett 15: 4230-4 (2005)
Article DOI: 10.1016/j.bmcl.2005.06.067 BindingDB Entry DOI: 10.7270/Q2ZG6RST |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 6
(Homo sapiens (Human)) | BDBM34142
(2-ethyl-5-methoxy-N,N-dimethyltryptamine | CHEMBL2...)Show InChI InChI=1S/C15H22N2O/c1-5-14-12(8-9-17(2)3)13-10-11(18-4)6-7-15(13)16-14/h6-7,10,16H,5,8-9H2,1-4H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 85 | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsson Research AB
Curated by ChEMBL
| Assay Description Inhibitory activity against 5-hydroxytryptamine 6 receptor in human |
Bioorg Med Chem Lett 15: 4230-4 (2005)
Article DOI: 10.1016/j.bmcl.2005.06.067 BindingDB Entry DOI: 10.7270/Q2ZG6RST |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human)) | BDBM34142
(2-ethyl-5-methoxy-N,N-dimethyltryptamine | CHEMBL2...)Show InChI InChI=1S/C15H22N2O/c1-5-14-12(8-9-17(2)3)13-10-11(18-4)6-7-15(13)16-14/h6-7,10,16H,5,8-9H2,1-4H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 620 | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsson Research AB
Curated by ChEMBL
| Assay Description Inhibitory activity against 5-hydroxytryptamine 2A receptor in human |
Bioorg Med Chem Lett 15: 4230-4 (2005)
Article DOI: 10.1016/j.bmcl.2005.06.067 BindingDB Entry DOI: 10.7270/Q2ZG6RST |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat)) | BDBM34142
(2-ethyl-5-methoxy-N,N-dimethyltryptamine | CHEMBL2...)Show InChI InChI=1S/C15H22N2O/c1-5-14-12(8-9-17(2)3)13-10-11(18-4)6-7-15(13)16-14/h6-7,10,16H,5,8-9H2,1-4H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsson Research AB
Curated by ChEMBL
| Assay Description Inhibitory activity against 5-hydroxytryptamine 1A receptor in rat |
Bioorg Med Chem Lett 15: 4230-4 (2005)
Article DOI: 10.1016/j.bmcl.2005.06.067 BindingDB Entry DOI: 10.7270/Q2ZG6RST |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 3A
(Homo sapiens (Human)) | BDBM34142
(2-ethyl-5-methoxy-N,N-dimethyltryptamine | CHEMBL2...)Show InChI InChI=1S/C15H22N2O/c1-5-14-12(8-9-17(2)3)13-10-11(18-4)6-7-15(13)16-14/h6-7,10,16H,5,8-9H2,1-4H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsson Research AB
Curated by ChEMBL
| Assay Description Inhibitory activity against 5-hydroxytryptamine 3 receptor expressed in NG 108 cells |
Bioorg Med Chem Lett 15: 4230-4 (2005)
Article DOI: 10.1016/j.bmcl.2005.06.067 BindingDB Entry DOI: 10.7270/Q2ZG6RST |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat)) | BDBM34142
(2-ethyl-5-methoxy-N,N-dimethyltryptamine | CHEMBL2...)Show InChI InChI=1S/C15H22N2O/c1-5-14-12(8-9-17(2)3)13-10-11(18-4)6-7-15(13)16-14/h6-7,10,16H,5,8-9H2,1-4H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsson Research AB
Curated by ChEMBL
| Assay Description Inhibitory activity against 5-hydroxytryptamine 1B receptor in rat |
Bioorg Med Chem Lett 15: 4230-4 (2005)
Article DOI: 10.1016/j.bmcl.2005.06.067 BindingDB Entry DOI: 10.7270/Q2ZG6RST |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human)) | BDBM34142
(2-ethyl-5-methoxy-N,N-dimethyltryptamine | CHEMBL2...)Show InChI InChI=1S/C15H22N2O/c1-5-14-12(8-9-17(2)3)13-10-11(18-4)6-7-15(13)16-14/h6-7,10,16H,5,8-9H2,1-4H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsson Research AB
Curated by ChEMBL
| Assay Description Inhibitory activity against 5-hydroxytryptamine 1D receptor in calf |
Bioorg Med Chem Lett 15: 4230-4 (2005)
Article DOI: 10.1016/j.bmcl.2005.06.067 BindingDB Entry DOI: 10.7270/Q2ZG6RST |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 7
(Homo sapiens (Human)) | BDBM34142
(2-ethyl-5-methoxy-N,N-dimethyltryptamine | CHEMBL2...)Show InChI InChI=1S/C15H22N2O/c1-5-14-12(8-9-17(2)3)13-10-11(18-4)6-7-15(13)16-14/h6-7,10,16H,5,8-9H2,1-4H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsson Research AB
Curated by ChEMBL
| Assay Description Inhibitory activity against 5-hydroxytryptamine 7 receptor in human |
Bioorg Med Chem Lett 15: 4230-4 (2005)
Article DOI: 10.1016/j.bmcl.2005.06.067 BindingDB Entry DOI: 10.7270/Q2ZG6RST |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human)) | BDBM34142
(2-ethyl-5-methoxy-N,N-dimethyltryptamine | CHEMBL2...)Show InChI InChI=1S/C15H22N2O/c1-5-14-12(8-9-17(2)3)13-10-11(18-4)6-7-15(13)16-14/h6-7,10,16H,5,8-9H2,1-4H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsson Research AB
Curated by ChEMBL
| Assay Description Inhibitory activity against 5-hydroxytryptamine 2C receptor in human |
Bioorg Med Chem Lett 15: 4230-4 (2005)
Article DOI: 10.1016/j.bmcl.2005.06.067 BindingDB Entry DOI: 10.7270/Q2ZG6RST |
More data for this Ligand-Target Pair | |