Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gamma-aminobutyric acid type B receptor subunit 1/2 (Homo sapiens (Human)) | BDBM50032964 ((R)-4-Amino-3-(4-chloro-phenyl)-butyric acid | 4-A...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
CIBA-GEIGY AG Curated by ChEMBL | Assay Description Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellum | J Med Chem 38: 3297-312 (1995) BindingDB Entry DOI: 10.7270/Q2N58KDP | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50032964 ((R)-4-Amino-3-(4-chloro-phenyl)-butyric acid | 4-A...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
CIBA-GEIGY AG Curated by ChEMBL | Assay Description Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortex | J Med Chem 38: 3297-312 (1995) BindingDB Entry DOI: 10.7270/Q2N58KDP | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50032964 ((R)-4-Amino-3-(4-chloro-phenyl)-butyric acid | 4-A...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Displacement of [3H]-GABA from Gamma-aminobutyric acid type B receptor | J Med Chem 42: 2053-9 (1999) Article DOI: 10.1021/jm990076+ BindingDB Entry DOI: 10.7270/Q2WW7GV9 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |