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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for UniProtKB: P25440   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Bromodomain-containing protein 2 [349-450]


(Homo sapiens (Human))
BDBM528580
PNG
(US11192900, Compound 3 | US11192900, Example S-10)
Show SMILES CNc1cc(cn(C)c1=O)-c1cc(NS(=O)(=O)C=C)ccc1Oc1ccc(F)cc1F
PDB
MMDB

Reactome pathway
KEGG

UniProtKB/SwissProt

B.MOAD
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 12n/an/an/an/an/an/a


TBA

Assay Description
The bromodomain binding assays were performed by Reaction Biology Corp., Malvern, Pa., USA (www.reactionbiology.com). The BET binding assays were con...


Citation and Details

BindingDB Entry DOI: 10.7270/Q2XS5ZJK
More data for this
Ligand-Target Pair